Drug class

PAH Agents- Endothelin Receptor Antagonists

PAH agents that are endothelin receptor antagonists comprise a therapeutic drug class indicated for the management of pulmonary arterial hypertension (WHO Group 1). Read more about PAH Agents- Endothelin Receptor Antagonists

35 drugs in this class 26 manufacturers

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Drugs in PAH Agents- Endothelin Receptor Antagonists

Showing 28–35 of 35 drugs

MACITENTAN

PAH AGENTS- ENDOTHELIN RECEPTOR ANTAGONISTS · PULMONARY ARTERIAL HYPERTENSION
Mylan Pharmaceuticals

MACITENTAN

PAH AGENTS- ENDOTHELIN RECEPTOR ANTAGONISTS · PULMONARY ARTERIAL HYPERTENSION
TEVA PHARM

MACITENTAN

PAH AGENTS- ENDOTHELIN RECEPTOR ANTAGONISTS · PULMONARY ARTERIAL HYPERTENSION
ALEMBIC PHARMAC

MACITENTAN

PAH AGENTS- ENDOTHELIN RECEPTOR ANTAGONISTS · PULMONARY ARTERIAL HYPERTENSION
APOTEX CORP

MACITENTAN

PAH AGENTS- ENDOTHELIN RECEPTOR ANTAGONISTS · PULMONARY ARTERIAL HYPERTENSION
ALEMBIC PHARMAC

MACITENTAN

PAH AGENTS- ENDOTHELIN RECEPTOR ANTAGONISTS · PULMONARY ARTERIAL HYPERTENSION
SANDOZ

MACITENTAN

PAH AGENTS- ENDOTHELIN RECEPTOR ANTAGONISTS · PULMONARY ARTERIAL HYPERTENSION
LAURUS LABS LIM

MACITENTAN

PAH AGENTS- ENDOTHELIN RECEPTOR ANTAGONISTS · PULMONARY ARTERIAL HYPERTENSION
ANI PHARMACEUTI
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About PAH Agents- Endothelin Receptor Antagonists.

PAH agents that are endothelin receptor antagonists comprise a therapeutic drug class indicated for the management of pulmonary arterial hypertension (WHO Group 1).

These agents—including ambrisentan, bosentan, and macitentan—function by competitively binding to and blocking endothelin receptors (ETA and/or ETB) on vascular smooth muscle cells.

By impeding the actions of endothelin-1, a potent endogenous vasoconstrictor and smooth muscle mitogen, they induce pulmonary vasodilation, attenuate abnormal vascular remodeling, improve exercise capacity, and reduce the risk of clinical disease progression.